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Publications During 2017

Sharma, R.; Gatchie, L.; Williams, I.S.; Jain, S. K.; Vishwakarma, R.A.; Chaudhuri, B.; Bharate, S. B. Glycyrrhiza glabra extract and quercetin reverses cisplatin resistance in triple-negative MDA-MB-468 breast cancer cells via inhibition of cytochrome P450 1B1 enzyme. Bioorganic & Medicinal Chemistry Letters ,2017, 27(24), 5400-5403.
Horley ,N. J.; Beresford, K.J .M; Kaduskar ,S.; McCann, G.J .P; Ruparelia, K.C; Sonawane ,V.R; Joshi, P.; Williams, I. S; Gatchie, L.; Bharate, S.B; et al. (E)-3-(3,4,5-Trimethoxyphenyl)-1-(pyridin-4-yl)prop-2-en-1-one, a heterocyclic chalcone is a potent and selective CYP1A1 inhibitor and cancer chemopreventive agent. Bioorganic & medicinal chemistry letters ,2017, 27(24), 5409-5414.
Jeelani, S.M.; Farooq, U.; Gupta, A.P.; Lattoo, S.K. Phytochemical evaluation of major bioactive compounds in different cytotypes of five species of Rumex L. Industrial Crops and Products ,2017, 109, 897-904. 
Singh, U.; Chashoo, G.; Khan, S. U.; Mahajan, P.; Nargotra, A.; Mahajan, G.; Singh, A.; Sharma, A.; Mintoo, M.J.; Guru, S.K.; et al. Design of Novel 3-Pyrimidinylazaindole CDK2/9 Inhibitors with Potent In Vitro and In Vivo Antitumor Efficacy in a Triple-Negative Breast Cancer Model. Journal of Medicinal Chemistry ,2017, 60(23), 9470-9489.
Borgohain, H.; Devi, R.; Dheer, D.; Borah, B.J.; Shankar, R.; Das, S.K. Synthesis of Tetrahydroquinoline-Embedded Bridged Benzothiaoxazepine-1,1-dioxides. European Journal Of Organic Chemistry ,2017,  (45), 6671-6679.
Rather, M.A.; Rasool, F.; Bhat, Z. S.; Dar, H.; Maqbool, M.; Amin, S.; Yousuf, S. K.; Ahmad, Z. Design and synthesis of indolopyridone hybrids as new antituberculosis agents. Microbial Pathogenesis ,2017, 113, 330-334.
Khan, S.; Kumar, A.; Gupta, R.; Ahmed, Q.N. The Ritter Reaction of 2-Oxoaldehydes at Room Temperature: Divergent Behaviour towards Acid Strength. ChemistrySelect ,2017, 2(34), 11336-11340.
Sharma, A.; Magotra, A.; Dogra, A.; Rath, S.K.; Rayees, S.; Wazir, P.; Sharma, S.; Sangwan, P.L.; Singh, S.; Singh, G.; Nandi, U. Pharmacokinetics, pharmacodynamics and safety profiling of IS01957, a preclinical candidate possessing dual activity against inflammation and nociception. Regulatory Toxicology and Pharmacology ,2017, 91, 216-225.
Arora, D.; Kumar, A.; Gupta, P.; Chashoo, G.; Jaglan, S. Preparation, characterization and cytotoxic evaluation of bovine serum albumin nanoparticles encapsulating 5-methylmellein: A secondary metabolite isolated from Xylaria psidii. Bioorganic & Medicinal Chemistry Letters ,2017, 27(23), 5126-5130.
Sharma, R.; Magotra, A.; Manhas, R.S.; Chaubey, A. Antagonistic potential of a psychrotrophic fungus: &ITTrichoderma velutinum&IT ACR-P1. Biological Control, 2017, 115, 12-17.
Kour, P.; Kumar, A.; Sharma, R.; Chib, R.; Khan, I.A.; Rai, V.K. Synthesis of 2-amino-4H-chromen-4-ylphosphonates and beta-phosphonomalonates via tandem Knoevenagel-Phospha-Michael reaction and antimicrobial. Research On Chemical Intermediates ,2017, 43(12), 7319-7329. 
Alam, N.; Koul, M.; Mintoo, M.J.; Khare, V.; Gupta, R.; Rawat, N.; Sharma, P. R.; Singh, S. K.; Mondhe, D. M.; Gupta, P. N. Development and characterization of hyaluronic acid modified PLGA based nanoparticles for improved efficacy of cisplatin in solid tumor. Biomedicine & Pharmacotherapy ,2017, 95, 856-864.
Bhat, Z. S.; Rather, M.A.; Maqbool, M.; Ul Lah, H.; Yousuf, S. K.; Ahmad, Z. Cell wall: A versatile fountain of drug targets in Mycobacterium tuberculosis. Biomedicine & Pharmacotherapy ,2017, 95, 1520-1534.
Kaur ,M. S.; Kaur ,R.; Bhatia, R.; Kumar ,K.; Kaur, R.; Singh, V.; Shankar, R.; Rawal, R. K. Synthetic and medicinal perspective of thiazolidinones: A review. Bioorganic chemistry , 2017, 75406-423.
Singh, G.; Razak, M.; Katoch, M.; Singh, G.; Katoch ,A.; Goswami ,A.; Katoch, M.; Katoch ,A.; Goswami, A.; Kitchlu ,S. Bioactive and biocontrol potential of endophytic fungi associated with Brugmansia aurea Lagerh. FEMS microbiology letters ,2017, 364(21).
By Bhat, Z. S.; Rather, M. A.; Syed, K.Y.; Ahmad, Z. α-pyrones and their hydroxylated analogs as promising scaffolds against Mycobacterium tuberculosis. Future Medicinal Chemistry, 2017, 9(17), 2053-2067.
Kumar, C.; Rasool, R.U.; Iqra, Z.; Nalli, Y.; Dutt, P.; Satti, N.K.; Sharma, N.; Gandhi, S.G.; Goswami, A.; Ali, A. Alkyne-azide cycloaddition analogues of dehydrozingerone as potential anti-prostate cancer inhibitors via the PI3K/Akt/NF-kappa B pathway. MedChemComm, 2017, 8(11), 2115-2124.
Rather, M. A.; Lone, A.M.; Teli, B.; Bhat, Z. S.; Singh, P.; Maqbool, M.; Shairgojray, B. A.; Dar, M. J.; Amin, S.; Yousuf, S.K.; et al. The synthesis, biological evaluation and structure-activity relationship of 2-phenylaminomethylene-cyclohexane-1,3-diones as specific anti-tuberculosis agents. MedChemComm ,2017, 8(11), 2133-2141, DOI:10.1039/C7MD00350A.
Kumar, S.; Nalli, Y.; Qadri, M.; Riyaz-Ul-Hassan, S.; Satti, N. K.; Gupta, V.; Bhushan, S.; Ali, A. Isolation of three new metabolites and intervention of diazomethane led to separation of compound 1 & 2 from an endophytic fungus, Cryptosporiopsis sp. depicting cytotoxic activity. Medicinal Chemistry Research ,2017, 26(11), 2900-2908.
Wani, N. A.; Singh, G.; Shankar, S.; Sharma, A.; Katoch, M.; Rai, R. Short hybrid peptides incorporating β- and γ-amino acids as antimicrobial agents. Peptides ,2017, 97, 46-53.
Ayoob, I.; Lone, S.H.; Masood-ur-R.; Zargar, O.A.; Bashir, R.; Shakeel-u-R.; Khuroo, M.A.; Bhat, K.A. New Semi-Synthetic Rosmarinic Acid-Based Amide Derivatives as Effective Antioxidants. CHEMISTRYSELECT ,2017, 2(31), 10153-10156.
Rasool, F.; Nayak D.; Katoch, A.; Faheem, M. M.; Yousuf ,S. K.; Hussain, N.; Goswami ,A.; Mukherjee ,D.; Rasool, F.; Hussain ,N.; et al. Regiospecific Synthesis of Ring A Fused Withaferin A Isoxazoline Analogues: Induction of Premature Senescence by W-2b in Proliferating Cancer Cells. Scientific reports ,2017, 7(1), 13749.
Kumar, V.; Gupta, M.; Gandhi, S. G.; Bharate, S.S.; Kumar, A.; Vishwakarma, R. A.; Bharate, S. B. Anti-inflammatory chromone alkaloids and glycoside from Dysoxylum binectariferum. Tetrahedron Letters ,2017, 58(42), 3974-3978. 
Singh, R.; Kumar, V.; Bharate, S. S.; Vishwakarma, R. A. Synthesis, pH dependent, plasma and enzymatic stability of bergenin prodrugs for potential use against rheumatoid arthritis. Bioorganic & Medicinal Chemistry ,2017, 25(20), 5513-5521.
Saneja, A.; Kumar, R.; Singh, A.; Dhar, D.R.; Mintoo, M. J.; Singh, G.; Mondhe, D. M.; Panda, A.K.; Gupta, P. N. Development and evaluation of long-circulating nanoparticles loaded with betulinic acid for improved anti-tumor efficacy. International Journal of Pharmaceutics (Amsterdam, Netherlands) ,2017, 531(1), 153-166.
Singh ,S.; Kalia ,N.P.; Khan ,I.A.; Singh, S.; Joshi, P.; Sharma ,P. R.; Kumar, A.; Bharate ,S. B.; Khan, I. A.; Joshi, P.; et al. Boeravinone B, A Novel Dual Inhibitor of NorA Bacterial Efflux Pump of Staphylococcus aureus and Human P-Glycoprotein, Reduces the Biofilm Formation and Intracellular Invasion of Bacteria. Frontiers in microbiology ,2017, 81868.
Rashid, S.; Bhat, B. A.; Mehta, G. Synthesis of pleurolactone and related mono- and sesquiterpenoids: Bioactive constituents of edible mushrooms. Tetrahedron Letters ,2017, 58(40), 3800-3802.
Sharma, R.; Abdullaha, M.; Bharate, S.B. Metal-Free Ionic-Liquid-Mediated Synthesis of Benzimidazoles and Quinazolin-4(3H)-ones from Benzylamines. Asian Journal of Organic Chemistry ,2017, 6(10), 1370-1374.
Shah, A.; Hassan, Q.P.; Mushtaq ,S.; Shah ,A. M.; Hussain ,A.; Shah ,A.; Hassan, Q. P.; Shah, A. M.; Hussain ,A. Chemoprofile and functional diversity of fungal and bacterial endophytes and role of ecofactors - A review. Journal of basic microbiology ,2017, 57(10), 814-826.
Chinthakindi, P.K.; Rath, S. K.; Singh, J.; Singh, S.; Koul, S.; Sangwan, P. L. Isolation of isoxanthanol and synthesis of novel derivatives as potential cytotoxic agents. Medicinal Chemistry Research ,2017, 26(10), 2499-2513.
Awasthi, P.; Singh, A.; Sheikh, G.; Mahajan, V.; Gupta, A.P.; Gupta, S.; Bedi, Y. S.; Gandhi, S. G. Mining and characterization of EST-SSR markers for Zingiber officinale Roscoe with transferability to other species of Zingiberaceae. Physiology and Molecular Biology of Plants ,2017, 23(4), 925-931.
Joshi, P.; Vishwakarma, R.A.; Bharate, S. B. Natural alkaloids as P-gp inhibitors for multidrug resistance reversal in cancer. European Journal of Medicinal Chemistry ,2017, 138, 273-292.
Jan ,A.T.; Rahman, S.; Yeo ,H.R.; Lee, E. J.; Choi ,I.; Malik ,M. A; Abdullah, T. S. Perspective Insights of Exosomes in Neurodegenerative Diseases: A Critical Appraisal. Frontiers in aging neuroscience ,2017,9317.
Sharma, S.; Kumar, A.; Mintoo ,M. J.; Mondhe, D. M.; Guru ,S. K.; Manda, S.; Bharate ,S. B. Prasad, V.D.; Sharma, P. R.; Bhushan ,S. A marine sponge alkaloid derivative 4-chloro fascaplysin inhibits tumor growth and VEGF mediated angiogenesis by disrupting PI3K/Akt/mTOR signaling cascade. Chemico-biological interactions,2017, 27547-60.
Sharma, R.; Abdullaha, M.; Bharate, S. B. Oxidant-Controlled C-sp2/sp3-H Cross-Dehydrogenative Coupling of N-Heterocycles with Benzylamines. Journal of Organic Chemistry ,2017, 82(18), 9786-9793.
Kumar, A.; Khan, S.; Ahmed, Q. N. Base-Controlled Reactions through an Aldol Intermediate Formed between 2-Oxoaldehydes and Malonate Half Esters. Organic Letters ,2017, 19(18), 4730-473.
Rasool, F.; Mukherjee, D. Pd-Catalyzed Regio- and Stereoselective C-Nucleoside Synthesis from Un-activated Uracils and Pyranoid Glycals. Organic Letters ,2017, 19(18), 4936-4939.
Singh ,H.; Singh ,J.V; Nepali, K.; Bedi, P. M. S; Gupta, M. K; Saxena, A. K; Sharma, S. Triazole tethered isatin-coumarin based molecular hybrids as novel antitubulin agents: Design, synthesis, biological investigation and docking studies. Bioorganic & medicinal chemistry letters ,2017, 27(17), 3974-3979.
Shah, A. M.; Shakeel,R.; Hussain, A.; Mushtaq, S.; Rather, M.A.; Shah, A.; Ahmad, Z.; Khan, I.A. ;Bhat, K.A.; Hassan, Q.P. Antimicrobial investigation of selected soil actinomycetes isolated from unexplored regions of Kashmir Himalayas, India. Microbial Pathogenesis ,2017, 110, 93-99.
Nissar, A. U.; Sharma, L.; Mudasir, M.A.; Nazir, L. A.; Umar, S. A.; Sharma, P.R.; Vishwakarma, R.A.; Tasduq, S. A. Chemical chaperone 4-phenyl butyric acid (4-PBA) reduces hepatocellular lipid accumulation and lipotoxicity through induction of autophagy. Journal of Lipid Research,2017, 58(9), 1855-186.
Pandith, S. A.; Dhar, N.; Wani, T.A.; Razdan, S.; Bhat, W. W.; Rana, S.; Khan, S.; Verma, M.K.; Lattoo, S.K. Production dynamics in relation to ontogenetic development and induction of genetic instability through in vitro approaches in Pelargonium graveolens: A potential essential oil crop of commercial significance.  Flavour and Fragrance Journal,2017, 32(5), 376-387.
Hussain, A.; Rather, M. A.; Shah, A. M.; Bhat, Z. S.; Shah, A.; Ahmad, Z.; Parvaiz Hassan, Q. Antituberculotic activity of actinobacteria isolated from the rare habitats. Letters in Applied Microbiology ,2017, 65(3), 256-264.
Rather, S. A.; Shah, A.M.; Ali, S. A.; Dar, R. A.; Rah, B.; Ali, A.; Hassan, Q. P. Isolation and characterization of Streptomyces tauricus from Thajiwas glacier-a new source of actinomycin-D. Medicinal Chemistry Research ,2017, 26(9), 1897-1902.
Dar, N. J.; Bhat, J. A.; Satti, N. K.; Sharma, P. R.; Hamid, A.; Ahmad, M. Withanone, an Active Constituent from Withania somnifera, Affords Protection Against NMDA-Induced Excitotoxicity in Neuron-Like Cells. Molecular Neurobiology ,2017, 54(7), 5061-5073.
Williams, I. S.; Gatchie, L.; Chaudhuri ,B.; Williams, I. S.; Gatchie, L.; Chaudhuri, B.; Chib ,S.; Saran, S.; Nuthakki ,V.K.; Joshi ,P.; et al. Biotransformation of Chrysin to Baicalein: Selective C6-Hydroxylation of 5,7-Dihydroxyflavone Using Whole Yeast Cells Stably Expressing Human CYP1A1 Enzyme. Journal of agricultural and food chemistry ,2017, 65(34), 7440-7446.
Kour, G.; Singh, P. ; Bhagat, A.; Ahmed, Z. Biopharmaceutic parameters, pharmacokinetics, transport and CYP-mediated drug interactions of IIIM-017: A novel nitroimidazooxazole analogue with anti-tuberculosis activity. European Journal of Pharmaceutical Sciences ,2017,106, 71-78.
Husain ,I.; Bala ,K.; Wani, A.; Makhdoomi ,U.; Malik ,F.; Sharma, A. Arginase purified from endophytic Pseudomonas aeruginosa IH2: Induce apoptosis through both cell cycle arrest and MMP loss in human leukemic HL-60 cells. Chemico-biological interactions , 2017, 27435-49.
Wani, Z. A.; Sultan, P.; Ashraf, N.; Wani, Z. A.; Riyaz-Ul-Hassan ,S.; Ashraf, N.; Kumar, A.; Bindu ,K.; Riyaz-Ul-Hassan ,S. Mortierella alpina CS10E4, an oleaginous fungal endophyte of Crocus sativus L. enhances apocarotenoid biosynthesis and stress tolerance in the host plant. Scientific reports , 2017, 7(1), 8598.
Magotra, A.; Sharma, A.; Gupta, A. P.; Wazir, P.; Sharma, S.; Singh, P. P.; Tikoo, M.K.; Vishwakarma, R. A.; Singh, G.; Nandi, U. Development and validation of a highly sensitive LC-ESI-MS/MS method for estimation of IIIM-MCD-211, a novel nitrofuranyl methyl piperazine derivative with potential activity against tuberculosis: Application to drug development. Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences ,2017, 1060, 200-206.
Williams, I. S.; Gatchie, L.; Joshi, P.; Vishwakarma ,R.A.; Sharma, M.; Satti ,N. K.; Chaudhuri ,B.; Bharate ,S. B. Synthesis and biological evaluation of pyrrole-based chalcones as CYP1 enzyme inhibitors, for possible prevention of cancer and overcoming cisplatin resistance. Bioorganic & medicinal chemistry letters , 2017, 27(16), 3683-3687.
Gupta, L.; Sharma, A. K.; Gothwal ,A.; Khan, M. S.; Khinchi, M. P.; Qayum, A.; Singh, S.K.; Gupta ,U. Dendrimer encapsulated and conjugated delivery of berberine: A novel approach mitigating toxicity and improving in vivo pharmacokinetics. International journal of pharmaceutics ,2017, 528(1-2), 88-99.
Kumar, S.; Kour, G.; Schreckenbach, G.; Andotra, S.; Hundal, G.; Sharma, V.; Jaglan, S.; Pandey, S.K. 3,4-Dimethyl diphenyldithiophosphate of mononuclear cobalt(II) with N-donor ligands: Synthesis, structural characterization, DFT and antibacterial studies. Journal of Molecular Structure ,2017, 1141, 23-30.
Koul,M.; Kumar, A.; Singh, J.; Sharma ,P. R.; Singh ,S.; Koul, M.; Kumar ,A.; Deshidi ,R.; Sharma ,V.; Singh ,J.; et al. Cladosporol A triggers apoptosis sensitivity by ROS-mediated autophagic flux in human breast cancer cells. BMC cell biology ,2017, 18(1), 26.
Katoch, M.; Singh, G.; Paul, A.; Sridhar ,S .N. C. Fungal endophytes associated with Viola odorata Linn. as bioresource for pancreatic lipase inhibitors. BMC complementary and alternative medicine ,2017, 17(1), 385.
Mahajan, P.; Chashoo, G.; Gupta, M.; Kumar, A.; Singh, P. P.; Nargotra, A. Fusion of Structure and Ligand Based Methods for Identification of Novel CDK2 Inhibitors. Journal of Chemical Information and Modeling ,2017, 57(8), 1957-1969.
Khajuria, V.; Gupta, S.; Sharma, N.; Kumar, A.; Lone, N.A.; Khullar, M.; Dutt, P.; Sharma, P. R. Bhagat, A.; Ahmed, Z. Anti-inflammatory potential of hentriacontane in LPS stimulated RAW 264.7 cells and mice model. Biomedicine & Pharmacotherapy ,2017, 92, 175-186.
Batarseh ,Y.S; Kaddoumi ,A.; Bharate ,S.S.; Kumar, V.; Kumar, A.; Vishwakarma ,R. A.; Bharate ,S. B. Crocus sativus Extract Tightens the Blood-Brain Barrier, Reduces Amyloid β Load and Related Toxicity in 5XFAD Mice. ACS chemical neuroscience ,2017, 8(8), 1756-1766.
Katoch, M.; Singh, A.; Singh, G.; Wazir, P.; Kumar, R. Phylogeny, antimicrobial, antioxidant and enzyme-producing potential of fungal endophytes found in Viola odorata. Annals of Microbiology (Heidelberg, Germany) ,2017, 67(8), 529-540.
Gupta, N.; Rath, S. K.; Singh, J.; Qayum, A.; Singh, S.; Sangwan, P.L. Synthesis of novel benzylidene analogues of betulinic acid as potent cytotoxic agents. European Journal of Medicinal Chemistry , 2017, 135, 517-530.
Dheer, D.; Rawal, R. K.; Singh, V.; Sangwan, P. L.; Das, P.; Shankar, R. β-CD/CuI catalyzed regioselective synthesis of iodo substituted 1,2,3-triazoles, imidazo[1,2-a]-pyridines and benzoimidazo[2,1-b]thiazoles in water and their functionalization. Tetrahedron ,2017, 73(30), 4295-4306.
Gupta, N.; Sharma, S.; Raina, A.; Bhushan, S.; Malik, F. A.; Sangwan, P. L. Synthesis of Novel Mannich Derivatives of Bakuchiol as Apoptotic Inducer through Caspase Activation and PARP-1 Cleavage in A549 Cells. ChemistrySelect ,2017, 2(18), 5196-5201.
Nageswar, R. D.; Rasheed, S.k.; Raina, G.; Ahmed, Q. N.; Jaladanki, C. K.; Bharatam, P.V.; Das, P. Cobalt-catalyzed regioselective ortho C(sp2)-H bond nitration of aromatics through proton-coupled electron transfer assistance. Journal of Organic Chemistry ,2017, 82(14), 7234-7244.
Anil, K. K.; Kannaboina, P.; Das, P. Ruthenium-catalyzed site-selective C-H arylation of 2-pyridones and 1-isoquinolinones. Organic & Biomolecular Chemistry,2017, 15(26), 5457-5461.
Sharma, R.; Jamwal, V.; Singh, V. P.; Wazir, P.; Awasthi, P.; Singh, D.; Vishwakarma, R.A.; Gandhi, S.G.; Chaubey, Asha. Revelation and cloning of valinomycin synthetase genes in Streptomyces lavendulae ACR-DA1 and their expression analysis under different fermentation and elicitation conditions. Journal of Biotechnology, 2017, 253, 40-47.
Dar ,M.S.; Singh ,P.; Mir, R. A.; Dar ,M. J. Βeta-catenin N-terminal domain: An enigmatic region prone to cancer causing mutations. Mutation research , 2017, 773122-133.
Bhat, Z.S.; Rather, M.r A.; Maqbool, M.; Lah, H. U. L.; Yousuf, S. K.; Ahmad, Z.. α-pyrones: Small molecules with versatile structural diversity reflected in multiple pharmacological activities-an update. Biomedicine & Pharmacotherapy ,2017, 91, 265-277.
Singh, J.; Qayum, A.; Singh, R. D.; Koul, M.; Kaul, A.; Satti, N. K.; Dutt, P.; Hamid, A.; Singh, S. Immunostimulatory activity of plumieride an iridoid in augmenting immune system by targeting Th-1 pathway in balb/c mice. International Immunopharmacology ,2017, 48, 203-210.
Nayak, D.; Kumar, A.; Chakraborty, S.; Rasool, R.; Amin, H.; Katoch, A.; Gopinath, V.; Mahajan, V.; Zilla, M. K.; Rah, B.l; et al. Inhibition of Twist1-mediated invasion by Chk2 promotes premature senescence in p53-defective cancer cells. Cell Death & Differentiation ,2017, 24(7), 1275-1287.
Dangroo, N. A.; Singh, J.; Rath, S. K.; Gupta, N.; Qayum, A.; Singh, S.; Sangwan, P. L. A convergent synthesis of novel alkyne-azide cycloaddition congeners of betulinic acid as potent cytotoxic agent. Steroids , 2017, 123, 1-12.
Wadhwa, B.; Makhdoomi, U.; Vishwakarma ,R.; Malik, F. Protein kinase B: emerging mechanisms of isoform-specific regulation of cellular signaling in cancer. Anti-cancer drugs , 2017, 28(6), 569-580.
Ramaraju, P.; Mir, N.A.; Singh, D.; Sharma, P.; Kant, R.; Kumar, I. An Unprecedented Pseudo-[3+2] Annulation between N-(4-Methoxyphenyl)aldimines and Aqueous Glutaraldehyde: Direct Synthesis of Pyrrole-2,4-dialdehydes. European Journal of Organic Chemistry, 2017, (24), 3461-3465.
Wani, T.A.; Pandith, S. A.; Gupta, A. P.; Chandra, S.; Sharma, N.; Lattoo, S. K. Molecular and functional characterization of two isoforms of chalcone synthase and their expression analysis in relation to flavonoid constituents in Grewia asiatica L. PLoS One ,2017, 12(6), e0179155/1-e0179155/24.
Gupta, A.; Kaur, R.; Singh, D.; Kapoor, K.K. Graphene oxide: A carbocatalyst for the one-pot multicomponent synthesis of highly functionalized tetrahydropyridines. Tetrahedron Letters,2017, 58(26), 2583-2587.
Nalli, Y.; Thakur, V.; Mohmmed, A.; Gupta, V.K.; Ali, A. POCl3-mediated cyclization of (+)-S-mahanimbine led to the divergent synthesis of natural product derivatives with antiplasmodial activity. New Journal of Chemistry ,2017, 41(12), 4923-4930.
Mehra, R.; Khan, I. A.; Nargotra, A. Anti-tubercular drug discovery: in silico implications and challenges. European Journal of Pharmaceutical Sciences ,2017, 104, 1-15.
Hudwekar, A. D.; Reddy, G. L.; Verma, P. K.; Gupta, S.; Vishwakarma, R. A.; Sawant, S. D. Transition Metal-free Single Step Approach for Arylated Pyrazolopyrimidinones and Quinazolinones Using Benzylamines/Benzylalcohols/Benzaldehydes. ChemistrySelect ,2017, 2(17), 4963-4968.
Andotra ,S.; Kumar, S.; Kour ,M.; Chayawan, V.; Sharma ,V.; Jaglan ,S.; Pandey, S.K. Synthesis, spectroscopic, DFT and in vitro biological studies of vanadium(III) complexes of aryldithiocarbonates. Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy , 2017, 180127-137.
Guleria, S.; Singh, G.; Gupta, S.; Vyas, D. Antioxidant and oxidative DNA damage protective properties of leaf, bark and fruit extracts of Terminalia chebula. Indian Journal of Biochemistry & Biophysics, 2017, 54(4), 127-134.
Katoch, M.; Bindu, K.; Phull, S.; Verma, M. K. An endophytic Fusarium sp isolated from Monarda citriodora produces the industrially important plant-like volatile organic compound hexanal. Microbiology (London, United Kingdom) ,2017, 163(6), 840-847.
Joshi, P.; Gupta, M.; Vishwakarma, R. A.; Kumar, A.; Bharate, S. B. (Z)-2-(3-Chlorobenzylidene)-3,4-dihydro-N-(2-methoxyethyl)-3-oxo-2H-benzo[b][1,4]oxazine-6-carboxamide as GSK-3β inhibitor: Identification by virtual screening and its validation in enzyme- and cell-based assay. Chemical Biology & Drug Design ,2017, 89(6), 964-971.
Krishnan, A.; Abdullah, T.S.; Mounajjed, T.; Hartono, S.; McConico, A.; White, T.; LeBrasseur, N.; Lanza, I.; Nair, S.; Gores, G.; Charlton, M. A longitudinal study of whole body, tissue, and cellular physiology in a mouse model of fibrosing NASH with high fidelity to the human condition. American journal of physiology. Gastrointestinal and liver physiology ,2017, 312(6), G666-G680.
Joshi, P.; McCann, G.J. P.; Sonawane, V. R.; Vishwakarma, R. A.; Chaudhuri, B. Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure-Based Virtual Screening and Their in Vitro Validation in Sacchrosomes and Live Human Cells. Journal of Chemical Information and Modeling ,2017, 57(6), 1309-1320, DOI:10.1021/acs.jcim.7b00095.
Hussain, A.; Rather, M. A.; Dar, M. S.; Aga, M. A.; Ahmad, N.; Manzoor, A.; Qayum, A.; Shah, A.; Mushtaq, S.; Ahmad, Z.; et al. Novel bioactive molecules from Lentzea violacea strain AS 08 using one strain-many compounds (OSMAC) approach. Bioorganic & Medicinal Chemistry Letters ,2017, 27(11), 2579-2582.
Malik, A. H.; Ashraf, N. Transcriptome wide identification, phylogenetic analysis, and expression profiling of zinc-finger transcription factors from Crocus sativus L. Molecular Genetics and Genomics ,2017, 292(3), 619-633.
Kumar, A.; Ahmed, Q.N. A Benzoquinone Imine Assisted Ring-Opening/Ring-Closing Strategy of the RCOCHN1N2 System: Dinitrogen Extrusion Reaction to Benzimidazoles. European Journal of Organic Chemistry ,2017, 2017(19), 2751-2756, DOI:10.1002/ejoc.201700357.
Das ,M.K.; Prajapati, B. K.; Ranjan ,K.; Tevatiya, S.; Sharma ,S.K.; Tiendrebeogo, R. W.; Kana, I. H.; Theisen, M.; Tiendrebeogo, R. W.; Kana ,I. H.; et al. Malaria epidemiology in an area of stable transmission in tribal population of Jharkhand, India. Malaria journal ,2017, 16(1), 181.
Rather, M.A.; Dar, B.A.; Shah, W.A.; Prabhakar, A.; Bindu, K.; Banday, J.A.; Qurishi, M.A. Comprehensive GC-FID, GC-MS and FT-IR spectroscopic analysis of the volatile aroma constituents of Artemisia indica and Artemisia vestita essential oils. Arabian Journal of Chemistry,2017, 10, S3798-S3803.
Rehman, S.; Latief, R.; Bhat, K.A.; Khuroo, M. A.; Shawl, A. S.; Chandra, S. Comparative analysis of the aroma chemicals of Melissa officinalis using hydrodistillation and HS-SPME techniques. Arabian Journal of Chemistry ,2017, 10(Suppl._2), S2485-S2490.
Rasool, R. U.; Nayak, D.; Chakraborty, S.; Faheem, M. M.; Rah, B.; Mahajan, P.; Gopinath, V.; Katoch, A.; Iqra, Z.; Yousuf, S. K.; et al. AKT is indispensable for coordinating Par-4/JNK cross talk in p21 downmodulation during ER stress. Oncogenesis ,2017, 6(5), e341.
Reddy, K. R.; Kannaboina, P.; Das, P. Palladium-Catalyzed Chemoselective Switch: Synthesis of a New Class of Indenochromenes and Pyrano[2,3-c]carbazoles. Asian Journal of Organic Chemistry ,2017, 6(5), 534-543.
Qadri, M.; Nalli, Y.; Jain, S. K.; Chaubey, A.; Ali, A.; Strobel, G.A.; Vishwakarma, R.A.; Riyaz-Ul-Hassan, S. An Insight into the Secondary Metabolism of Muscodor yucatanensis: Small-Molecule Epigenetic Modifiers Induce Expression of Secondary Metabolism-Related Genes and Production of New Metabolites in the Endophyte. Microbial Ecology ,2017, 73(4), 954-965.
Shah, A.; Rather, M. A.; Hassan, Q. P.; Aga, M. A.; Mushtaq, S.; Shah, A. M.; Hussain, A.; Baba, S. A.; Ahmad, Z. Discovery of anti-microbial and anti-tubercular molecules from Fusarium solani: an endophyte of Glycyrrhiza glabra. Journal of Applied Microbiology ,2017, 122(5), 1168-1176.
Ahmad, M.; Aga, M. A.; Bhat, J. A.; Kumar, B.; Rouf, A.; Capalash, N.; Mintoo, M.J.; Kumar, A.; Mahajan, P.; Mondhe, D. M.; et al. Exploring Derivatives of Quinazoline Alkaloid L-Vasicine as Cap Groups in the Design and Biological Mechanistic Evaluation of Novel Antitumor Histone Deacetylase Inhibitors. Journal of Medicinal Chemistry ,2017, 60(8), 3484-3497.
Siddique, M. ; Usman, M.; Jayaprakash ,V.; Sinha ,B. N.; McCann ,G. J .P.; Sonawane, V. R.; Horley, N.; Gatchie, L.; Joshi ,P.; Bharate ,S. B.; Chaudhuri, B. Quinazoline derivatives as selective CYP1B1 inhibitors. European journal of medicinal chemistry ,2017, 130320-327.
Ayoob, I.; Hazari, Y.M.; Lone, S.H.; Rehman ,S.; Khuroo, M.A.; Fazili, K.M.; Bhat, K.A. Phytochemical and Cytotoxic Evaluation of Peganum Harmala: Structure Activity Relationship Studies of Harmine. CHEMISTRYSELECT ,2017, 2(10), 2965-2968.
Singh, D.; Kumar, V.; Devi, N.; Malakar, C.C.; Shankar, R.; Singh, V. Metal-free Decarboxylative Amination: An Alternative Approach Towards Regioselective Synthesis of beta-Carboline N-fused Imidazoles. Advanced Synthesis & Catalysis,2017, 359(7), 1213-1226.
Thotakura, N.; Dadarwal, M.; Kumar ,P.; Raza, K.; Sharma ,G.; Katare ,O. P.; Guru, S. K.; Bhushan, S. Chitosan-Stearic Acid Based Polymeric Micelles for the Effective Delivery of Tamoxifen: Cytotoxic and Pharmacokinetic Evaluation. AAPS PharmSciTech ,2017, 18(3), 759-768.
Dheer ,D.; Singh ,V.; Shankar, R. Medicinal attributes of 1,2,3-triazoles: Current developments. Bioorganic chemistry ,2017, 7130-54.
Rather, L.J.; Akhter, S.; Padder, R.A.; Hassan, Q.P.; Hussain, M.; Khan, M.A.; Mohammad, F. Colorful and semi durable antioxidant finish of woolen yarn with tannin rich extract of Acacia nilotica natural dye. Dyes and Pigments,2017, 139, 812-819.
Saneja, A.; Sharma, L.; Singh, A.; Dubey, R. D.; Mintoo ,M.J.; Kumar, A.; Sangwan, P. L.; Abdullah, T. S.; Singh ,G,; Mondhe, D, M,; et al. Synthesis, characterization and augmented anticancer potential of PEG-betulinic acid conjugate. Materials science & engineering. C, Materials for biological applications ,2017, 73616-626.
Horley ,N. J.; Beresford ,K.J. M.; Chawla ,T.; McCann ,G. J. P.; Ruparelia, K.C; Sonawane ,V. R.; Tan, H. L.; Gatchie ,L.; Williams ,I. S.; Joshi, P.; et al. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines. European journal of medicinal chemistry ,2017, 129159-174.
Baba, S. A.; Vishwakarma, R.A.; Ashraf, N. Functional Characterization of CsBGlu12, a β-Glucosidase from Crocus sativus, Provides Insights into Its Role in Abiotic Stress through Accumulation of Antioxidant Flavonols. Journal of Biological Chemistry ,2017, 292(11), 4700-4713.
Katoch, M.; Phull ,S.; Vaid, S.; Singh ,S. uiversity, Phylogeny, anticancer and antimicrobial potential of fungal endophytes associated with Monarda citriodora L. BMC microbiology ,2017, 17(1), 44.
Ur Rasool, R.; Debasis, N.; Chakraborty, S.; Jamwal, V.L.; Mahajan, V.; Katoch, A.; Faheem, M. M..; Iqra, Z.; Amin, H.; Gandhi, S. G.; et al. Differential regulation of NM23-H1 under hypoxic and serum starvation conditions in metastatic cancer cells and its implication in EMT. European Journal of Cell Biology ,2017, 96(2), 164-171.
Dutta, S.; Godara ,R.; Katoch ,R.; Yadav ,A.; Katoch ,M.; Singh, N .K. Detection of amitraz and malathion resistance in field populations of Rhipicephalus (Boophilus) microplus (Acari: Ixodidae) in Jammu region of India. Experimental & applied acarology , 2017, 71(3), 291-301.
Singh, K.S.; Wang, P.; Narkhede, N.A.; Mozharivskyj, Y. Iridium(III) and Rhodium(III) compounds of dipyridyl-N-alkylimine and dipyridyl-NH-ketimine: Spectral characterization and crystal structure. Journal of Chemical Sciences ,2017, 129(3), 365-372.
Singh ,A.; Arvinda, S.; Suri ,J.; Singh ,S.; Koul, S.; Vishwakarma ,R.; Mondhe ,D. M.; Singh, G. IN0523 (Urs-12-ene-3α,24β-diol) a plant based derivative of boswellic acid protect Cisplatin induced urogenital toxicity. Toxicology and applied pharmacology , 2017, 3188-15.
Kumar, A.; Sharma, P. R.; Mondhe, D. M. Potential anticancer role of colchicine-based derivatives: an overview. Anti-Cancer Drugs ,2017, 28(3), 250-262.
Gurmeen, R.; Gobind, R.; Kaur, T.; Vyas, D.; Sharma, A. D.; Singh, J. Molecular cloning, characterization, heterologous expression and in-silico analysis of disordered boiling soluble stress-responsive wBsSRP protein from drought tolerant wheat cv.PBW 175. Plant physiology and biochemistry : PPB , 2017, 11229-44.
Magotra, A.; Kumar, M.; Kushwaha, M.; Awasthi, P.; Raina, C.; Gupta, A. P.; Shah, B. A.; Gandhi, S. G.; Chaubey, Asha. Epigenetic modifier induced enhancement of fumiquinazoline C production in Aspergillus fumigatus (GA-L7): an endophytic fungus from Grewia asiatica L. AMB Express , 2017, 7(1), 1-10.
Aga, M. A.; Rayees, S.; Rouf, A.; Kumar, B.; Sharma, A.; Nagaraju, P. V. V. S.; Singh, G.; Taneja, S.C. Synthesis of Ofornine mimics from natural product l-vasicine as anti-hypertensive agents. Bioorganic & Medicinal Chemistry ,2017, 25(4), 1440-1447.
Singh, G.; Singh ,G.; Bhatti ,R.; Gupta, V.; Mahajan ,A.; Singh, P.; Singh, I.M. P. Rationally designed benzopyran fused isoxazolidines and derived β(2,3,3)-amino alcohols as potent analgesics: Synthesis, biological evaluation and molecular docking analysis. European journal of medicinal chemistry ,2017, 127210-222.
Chinthakindi, P.K.; Singh, J.; Gupta, S.; Nargotra, A.; Mahajan, P.; Kaul, A.; Ahmed, Z.; Koul, S.; Sangwan, P.L. Synthesis of a-santonin derivatives for diminutive effect on T and B-cell proliferation and their structure activity relationships. European Journal of Medicinal Chemistry , 2017, 127, 1047-1058.
Gopalakrishna, P.;Geetha, K.; Bharate ,S.S.; Vishwakarma, R. A.; Awasthi ,A.; Verma ,R.; Mishra, G.; Singh, A. T.; Jaggi, M.; Mithal ,A. Antidiabetic potential of polyherbal formulation DB14201: Preclinical development, safety and efficacy studies. Journal of ethnopharmacology ,2017, 197218-230.
Devi ,P.; Wahidullah ,S.; Sheikh, F.; Pereira, R.; Amonkar, D.; Tilvi ,S.; Meena, R. M.; Narkhede Niteen. Biotransformation and Detoxification of Xylidine Orange Dye Using Immobilized Cells of Marine-Derived Lysinibacillus sphaericus D3. Marine drugs ,2017, 15(2).
Khan ,M. F.; Alam ,M. M.; Verma, G.; Akhtar, W.; Akhter ,M.; Shaquiquzzaman, M.; Rizvi ,M. A.; Ali, A. Molecular interactions of dioxins and DLCs with the ketosteroid receptors: an in silico risk assessment approach. Toxicology mechanisms and methods ,2017, 27(2), 151-163.
Dhamale, O.P.; Lawrence, R.; Wiegmann, E.M.; Shah, B.A.; Al-Mafraji, K.; Lamanna, W.C.; Lubke, T.; Dierks, T.; Boons, G.J.; Esko, J.D. Arylsulfatase K is the Lysosomal 2-Sulfoglucuronate Sulfatase. ACS Chemical Biology, 2017, 12(2), 367-373.
Rahat, B.; Kaur ,J.; Najar ,R.A.; Hamid, A.; Bagga ,R. The role of aberrant methylation of trophoblastic stem cell origin in the pathogenesis and diagnosis of placental disorders. Prenatal diagnosis ,2017, 37(2), 133-143.
Masood, R.; Mohammad ,Y.; Fazili ,K. M.; Bhat, K. A.; Ara, T. Synthesis and biological evaluation of novel 3-O-tethered triazoles of diosgenin as potent antiproliferative agents. Steroids , 2017, 1181-8.
Yedukondalu, N.; Arora, P.; Wadhwa, B.; Malik, F.A.; Vishwakarma, R.A.; Gupta, V. K.; Riyaz-Ul-Hassan, S.; Ali, A. Diapolic acid A-B from an endophytic fungus, Diaporthe terebinthifolii depicting antimicrobial and cytotoxic activity. Journal of Antibiotics ,2017, 70(2), 212-215.
Reddy, A. S.; Ranjith ,R.K.; Nageswar, R. D.; Jaladanki, C.K.; Bharatam, P.; Lam, P. Y. S.; Das, P. Copper(II)-catalyzed Chan-Lam cross-coupling: chemoselective N-arylation of aminophenols. Organic & Biomolecular Chemistry ,2017, 15(4), 801-806.
Mubashir, K.; Ganai, B. A.; Tantry, M.; Ghazanfar ,K.; Akbar, S.; Rah, B.; Masood, A. Anti-inflammatory and immuno-modulatory studies on LC-MS characterised methanol extract of Gentiana kurroo Royle. BMC complementary and alternative medicine ,2017, 17(1), 78.
Ravi ,C.; Chandra, M. D.; Qayum, A.; Singh ,S. K; Adimurthy ,S. Design, synthesis and cytotoxicity studies of novel pyrazolo[1, 5-a] pyridine derivatives. European journal of medicinal chemistry ,2017, 126277-285.
Yadav ,P.; Lal, K.; Kumar, A.; Guru, S. K.; Jaglan ,S.; Bhushan, S. Green synthesis and anticancer potential of chalcone linked-1,2,3-triazoles. European journal of medicinal chemistry ,2017, 126944-953.
Aruri, H.; Singh, U.; Kumar, M.; Sharma, S.; Aithagani, S. K.; Gupta, V. K.; Mignani, S.e; Vishwakarma, R.A.; Singh, P. Pal. Metal-free Cross-Dehydrogenative Coupling of HN-azoles with α-C(sp3)-H Amides via C-H Activation and Its Mechanistic and Application Studies. Journal of Organic Chemistry ,2017, 82(2), 1000-1012.
Rahat, B.; Mahajan ,A.; Kaur ,J.; Bagga ,R.; Hamid, A. Epigenetic modifications at DMRs of placental genes are subjected to variations in normal gestation, pathological conditions and folate supplementation. Scientific reports ,2017, 740774.
Borkar, S.R.; Bokolia, N.; Aidhen, I.S.; Khan, I.A. Synthesis of threo- and erythro-configured trihydroxy open chain lipophilic ketones as possible anti-mycobacterial agents. Tetrahedron-Asymmetry ,2017, 28(1).
Saneja, A.; Nayak ,D.; Srinivas, M.; Kumar ,A.; Khare, V.; Katoch ,A.; Goswami ,A.; Vishwakarma ,R. A; Sawant ,S. D.; Gupta, P. N. Development and mechanistic insight into enhanced cytotoxic potential of hyaluronic acid conjugated nanoparticles in CD44 overexpressing cancer cells. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences ,2017, 9779-91.
Dash, A.K.; Madhubabu, T.; Yousuf, S. K.; Raina, S.; Mukherjee, D. One-pot Mukaiyama type carbon-Ferrier rearrangement of glycals: Application in the synthesis of chromanone 3-C-glycosides. Carbohydrate Research ,2017, 438, 1-8.
Deshidi, R.; Devari, S.; Kushwaha, M.; Gupta, A.P.; Sharma, R.; Chib, R.; Khan, I.A.; Jaglan, S.; Shah, B.A. Isolation and Quantification of Alternariols from Endophytic Fungus, Alternaria alternata: LC-ESI-MS/MS Analysis. Chemistryselect ,2017, 2(1), 364-368.
Kour, M.; Kumar, S.; Andotra, S.; Kour, G.; Singh, G.; Gupta, V.K.; Kant, R.; Katoch, M.; Pandey, S.K. Chromium(III) complexes of dimethyl diphenyldithiophosphates: Synthesis, characterization, and antibacterial studies. Phosphorus Sulfur and Silicon and the Related Elements,2017, 192(10), 1119-1123.
Sharma, R; Khan, I. A. Mechanism and Potential Inhibitors of GlmU: A Novel Target for Antimicrobial Drug Discovery. Current Drug Targets ,2017,18(14), 1587-1597.
Dheer, D.; Reddy, K.R.; Rath, S.K.; Sangwan, P.L.; Das, P.; Shankar, R. Cu(I)-catalyzed double C-H amination: synthesis of 2-iodo-imidazo[1,2-a]pyridines . RSC Advances,2017, 7(64), 40591-40591.
Theisen ,M.; Adu, B.; Mordmuller, B.; Singh ,S. The GMZ2 malaria vaccine: from concept to efficacy in humans. Expert review of vaccines ,2017, 16(9), 907-917.
Nalli, Y.; Gupta, S.; Khajuria, V.; Singh, V. P.; Sajgotra, M.; Ahmed, Z.; Thakur, N. L.; Ali, A. TNF-α and IL-6 inhibitory effects of cyclic dipeptides isolated from marine bacteria Streptomyces sp. Medicinal Chemistry Research ,2017, 26(1), 93-100, DOI:10.1007/s00044-016-1730-8.
Valdiani, A.; Maziah ,M.; Abiri, R.; Talei, D.; Lattoo, S.r K.; Ortiz, R.; Rasmussen ,S.K.; Batley Jacqueline; Rafii Mohd Yusop; Maziah Mahmood; et al. Genoproteomics-assisted improvement of Andrographis paniculata: toward a promising molecular and conventional breeding platform for autogamous plants affecting the pharmaceutical industry. Critical reviews in biotechnology ,2017, 37(6), 803-816.
Khera, H.K.; Singh, S. K.; Mir, R.; Bharadwaj, V.; Singh, S. A HR-MS Based Method for the Determination of Chorismate Synthase Activity. Protein & Peptide Letters ,2017, 24(3), 229-234.
Katoch, M.; Pull ,S. Endophytic fungi associated with Monarda citriodora, an aromatic and medicinal plant and their biocontrol potential. Pharmaceutical biology ,2017, 55(1), 1528-1535.
Khare, V.; Al Sakarchi, W.; Gupta, P.N.; Curtis, A.D.M.; Hoskins, C. Synthesis and characterization of TPGS-gemcitabine prodrug micelles for pancreatic cancer therapy. RSC Advances,2017, 7(28), 17367-17367.
Sharma, S.; Gupta, M.K.; Saxena, A.K.; Bedi, P.M.S. Thiazolidinone Constraint Combretastatin Analogs as Novel Antitubulin Agents: Design, Synthesis, Biological Evaluation and Docking Studies. Anti-Cancer Agents in Medicinal Chemistry ,2017, 17(2), 230-240.
Shukla ,G.; Khare, P.; Patidar, R.; Saxena ,R.; Khera ,H. K.; Srivastava ,A. K. Therapeutic Potential, Challenges and Future Perspective of Cancer Stem Cells in Translational Oncology: A Critical Review. Current stem cell research & therapy ,2017, 12(3), 207-224.
Dheer,D.; Arora, D.; Jaglan ,S.; Shankar, R.; Dheer, D.; Shankar ,R.; Arora, D.; Jaglan, S.; Rawal, R. K. Polysaccharides based nanomaterials for targeted anti-cancer drug delivery. Journal of drug targeting ,2017, 25(1), 1-16.
Naseer, S.; Bhat, K. A.; Qadri, M.; Riyaz-Ul-Hassan, S.; Malik, F. A.; Khuroo, M. A. Bioactivity-guided isolation, antimicrobial and cytotoxic evaluation of secondary metabolites from Cladosporium tenuissimum associated with Pinus wallichiana. ChemistrySelect ,2017, 2(3), 1311-1314.
Singh V.; Singh B.; Sharma A.; Kaur K.; Pati P .K.; Gupta A. P.; Salar R. K.; Hallan V. Leaf spot disease adversely affects human health-promoting constituents and withanolide biosynthesis in Withania somnifera (L.) Dunal. Journal of applied microbiology ,2017, 122(1), 153-165.
Dangroo, N.A.; Singh, J.; Gupta, N.; Singh, S.; Kaul, A.; Khuroo, M.A.; Sangwan, P. T- and B-cell immunosuppressive activity of novel alpha-santonin analogs with humoral and cellular immune response in Balb/c mice. Medchemcomm,2017, 8(1), 211-219.
Kumar, B.; Singh, V.; Shankar, R.; Kumar, K.; Rawal, R.K. Synthetic and Medicinal Prospective of Structurally Modified Curcumins. Current Topics in Medicinal Chemistry  ,2017, 17(2), 148-161.
Mushtaq, S.; Hassan, Q.P.; Sharma, R.; Majeed, R.; Dar, A.H.; Sultan, P.; Khan, I.A.; Ali, S.A.; Ali, M.N. Evaluation of anticancer and antimicrobial activities of selected medicinal plants of Kashmir Himalayas, India. Indian Journal of Traditional Knowledge, 2017, 16(1), 141-145.
Razdan, S.; Bhat, W.W.; Dhar, N.; Rana, S.; Pandith, S.A.; Wani, T. A.; Vishwakarma, R.; Lattoo, S. K. Molecular characterization of DWF1 from Withania somnifera (L.) Dunal: its implications in withanolide biosynthesis. Journal of Plant Biochemistry and Biotechnology ,2017, 26(1), 52-63.
Mahajan, P.; Suri, N.; Mehra, R.; Gupta, M.; Kumar, A.; Singh, S. K.; Nargotra, A. Discovery of novel small molecule EGFR inhibitory leads by structure and ligand-based virtual screening. Medicinal Chemistry Research ,2017, 26(1), 74-92.
Malik ,T.A.; Kamili ,A. N.; Chishti ,M .Z.; Tantry ,M. A.; Ahad ,S.; Hussain, P. R.; Johri, R .K. Breaking the resistance of Escherichia coli: Antimicrobial activity of Berberis lycium Royle. Microbial pathogenesis , 2017, 10212-20.
Koul, M.; Singh, S. Penicillium spp.: prolific producer for harnessing cytotoxic secondary metabolites. Anti-Cancer Drugs , 2017, 28(1), 11-30.
Lone, M.I.; Nabi, A.; Dar ,N. J.; Hussain, A.; Nazam, N.; Ahmad, W.; Hamid ,A. Toxicogenetic evaluation of dichlorophene in peripheral blood and in the cells of the immune system using molecular and flow cytometric approaches. Chemosphere ,2017, 167520-529.
Rather, G. A.; Sharma, A.; Pandith, S. A.; Kaul, V.; Nandi, U.; Misra, P.; Lattoo, S. K. De novo transcriptome analyses reveals putative pathway genes involved in biosynthesis and regulation of camptothecin in Nothapodytes nimmoniana (Graham) Mabb. Plant Molecular Biology ,2017.
Gupta, S.; Ul Ahsan, A.; Wani, A.; Khajuria, V.; Nazir, L. A.; Sharma, S.; Bhagat, A.; Raj ,S.P.; Bhardwaj, S.; Peerzada, K. J.; et al. The amino analogue of β-boswellic acid efficiently attenuates the release of pro-inflammatory mediators than its parent compound through the suppression of NF-κB/IκBα signalling axis. Cytokine+, 2017, DOI:10.1016/j.cyto.2017.12.004.
Shankar, S.; Faheem, M. M.; Nayak, D.; Wani, N. A.; Farooq, S.; Koul, S.; Goswami, A.; Rai, R. Cyclodipeptide c(Orn-Pro) Conjugate with 4-Ethylpiperic Acid Abrogates Cancer Cell Metastasis through Modulating MDM2. Bioconjugate Chemistry ,2017,  DOI:10.1021/acs.bioconjchem.7b00670.
Bhat, Z. S.; Ul Lah, H.; Rather, M.A.; Maqbool, M.; Ara, T.; Ahmad, Z.; Yousuf, S. K. Synthesis and in vitro evaluation of substituted 3-cinnamoyl-4-hydroxy-pyran-2-one (CHP) in pursuit of new potential antituberculosis agents. MedChemComm ,2017, DOI:10.1039/c7md00366h.
Pandey, A. Bani, S.; Dutt, P.; Satti, Naresh .; Avtar, S.K.; Qazi, G. N. Multifunctional neuroprotective effect of Withanone, a compound from Withania somnifera roots in alleviating cognitive dysfunction. Cytokine+, 2017, DOI:10.1016/j.cyto.2017.10.019.
Wani, T. A.; Lattoo, S.K. Auxin response factor (GaARF) cloning and expression in relation to reproductive maturation in Grewia asiatica L. Plant Gene ,2017, 12, 123-130.
Sultan, S.; Gupta, V.; Shah, B. A. Photoredox-Catalyzed Isatin Reactions: Access to Dibenzo-1,7-Naphthyridine Carboxylate and Tryptanthrin. ChemPhotoChem ,2017, 1(4), 120-124.
Arora, D.; Jaglan, S. Therapeutic applications of resveratrol nanoformulations. Environmental Chemistry Letters ,2017, DOI:10.1007/s10311-017-0660-0.
Sharma, A.; Magotra, A.; Rath, S.K.; Wazir, P.; Nandi, U.; Koul, S.; Sangwan, P. L; Gupta, A. P.; Singh, G. In-vitro and in-vivo pharmacokinetics of IS01957, p-coumaric acid derivative using a validated LC-ESI-MS/MS method in mice plasma. Journal of Pharmaceutical Investigation ,2017, DOI:10.1007/s40005-017-0350-8.
Wani, N. A.; Raghothama, S.; Singh, U. P.; Rai, R. C11/C9 Helical folding in αβ hybrid peptides containing 1-amino-cyclohexane acetic acid (β3, 3-Ac6c). Chemistry - A European Journal ,2017, 23(35), 8364-8370.
Dar, N. J.; Satti, N. K.; Dutt, P.; Hamid, A.; Ahmad, M.. Attenuation of Glutamate-Induced Excitotoxicity by Withanolide-A in Neuron-Like Cells: Role for PI3K/Akt/MAPK Signaling Pathway. Molecular Neurobiology ,2017,  DOI:10.1007/s12035-017-0515-5.
Vishwakarma, R. Editorial: Medicinal Chemistry Research in India. ACS Medicinal Chemistry Letters ,2017, 8(3), 270-272.
Lone, S. H.; Rehman, S. U.; Bhat, K. A. Synthesis of Gallic-Acid-1-Phenyl-1H-[1,2,3]Triazol-4-yl Methyl Esters as Effective Antioxidants. Drug Research (Stuttgart, Germany) ,2017, 67(2), 111-118.
Arora ,D.; Sharma ,N.; Jaglan, S.; Arora ,D.; Sharma, N.; Chashoo ,G.; Singamaneni, V.; Gupta ,P. Bacillus amyloliquefaciens induces production of a novel blennolide k in co-culture of Setophoma terrestris. Journal of applied microbiology , 2017.
Dheer ,D.; Jyoti; Gupta ,P.N; Shankar, R. Tacrolimus: An updated review on delivering strategies for multifarious diseases. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences ,2017,  114217-227.
Mushtaq, S.; Shah ,A. M.; Shah, A.; Lone, S.A.; Hussain ,A.; Hassan, Q. P.; Ali ,M.N. Bovine mastitis: An appraisal of its alternative herbal cure. Microbial pathogenesis ,2017, 114357-361.
Najar, R.A.; Bhat ,J. A.; Dar ,N. J.; Wani, N. A.; Rahat, B.; Kaur, J.; Gupta, A.P.; Kaur ,J.; Hamid, A. Modulation of dietary folate with age confers selective hepatocellular epigenetic imprints through DNA methylation. The Journal of nutritional biochemistry ,2017, 53121-132.
Singh ,I.; Verma, V.; Chandra ,R.; Singh, I.; Verma ,V.; Singh, S.; Uversky ,V. N.; Uversky ,V.N. In silico evaluation of the resistance of the T790M variant of epidermal growth factor receptor kinase to cancer drug Erlotinib. Journal of biomolecular structure & dynamics ,2017, 1-11.
Magotra ,A.; Sharma, A.; Singh ,S.; Kumar ,S.; Ojha ,P. K.; Bokolia, N.; Khan, I. A.; Wazir, P.; Sharma, S.; Singh, P.P.; et al. Physicochemical, pharmacokinetic, efficacy and toxicity profiling of a potential nitrofuranyl methyl piperazine derivative IIIM-MCD-211 for oral tuberculosis therapy via in-silico-in-vitro-in-vivo approach. Pulmonary pharmacology & therapeutics ,2017.
Sharma, V.; Dhar ,M.K; Kaul ,S.; Kapoor, K.K.; Mukherjee ,D.; Gupta, V. K. Camphor sulphonic acid mediated quantitative 1,3-diol protection of major Labdane diterpenes isolated from Andrographis paniculata. Natural product research ,2017, 1-9.
Singh ,I.; Singh ,G.; Verma ,V; Chandra ,R.; Singh, I.; Verma ,V.; Singh, G.; Singh ,S. In Silico Evaluation of Variable pH on the Binding of Epidermal Growth Factor Receptor Ectodomain to its Ligand Through Molecular Dynamics Simulation in Tumors. Interdisciplinary sciences, computational life sciences ,2017.
Dubey ,R. D.; Gupta ,P.N.; Klippstein ,R.; Wang ,J. T.; Hodgins, N.; Mei Kuo,C.; Hider, R. C.; Abbate, V.; Al-Jamal Khuloud ,T.; Sosabowski ,J. Novel Hyaluronic Acid Conjugates for Dual Nuclear Imaging and Therapy in CD44-Expressing Tumors in Mice In Vivo. Nanotheranostics ,2017, 1(1), 59-79.
Kumar ,D.; Singh, G.; Bedi ,P.; Jain, S. K.; Sharma ,P.; Qayum ,A.; Mahajan ,G.; Mintoo ,M. J.; Singh ,S.K.; Mondhe, D. M.; et al. 4-aryl/heteroaryl-4H-fused pyrans as Anti-proliferative Agents: Design, Synthesis and Biological Evaluation. Anti-cancer agents in medicinal chemistry ,2017.
Kancherla ,P.; Alegete, P.; Khagga ,M.; Kancherla ,P.; Keesari ,S.; Alegete, P.; Das ,P. Identification, isolation, and synthesis of seven novel impurities of anti-diabetic drug Repaglinide. Drug testing and analysis ,2017.